Timoptic XE®

Timolol Maleate 0.25% or 0.5%
ophthalmic gel forming solution
Antiglaucoma
[ Non-selective beta-adrenergic receptor blocker]
Indication

Indication

Elevated intraocular pressure in ocular hypertension or open-angle glaucoma
Mechanism of Action

Mechanism of Action

Reduces aqueous formation by blocking beta2 receptors on nonpigmented ciliary epithelium. Reduces elevated and normal intraocular pressure.
Common quantities available

Available Quantities

2.5 ml, 5 ml
Dosage

Dosage/Instructions

1 drop 0.25% or 0.5% every morning
Pregnancy & Nursing Data

Pregnancy & Nursing

Increased fetal resorptions in rabbits at high doses. Use only if the potential benefit justifies the potential risk to the fetus.
Pediatric Use

Pediatric Use

No studies
Warnings Tab

Contraindications, side effects, etc.

Contraindicated in asthma, severe COPD, sinus bradycardia, heart block greater than first degree, cardiac failure, cardiogenic shock. Warnings include systemic absorption, cardiac failure, vascular insufficiency, obstructive pulmonary disease, diabetes mellitus, thyrotoxicosis, choroidal detachment. Adverse reactions: ocular burning, stinging, blepharoconjunctivitis, heart rate and blood pressure decrease, iridocyclitis, headache, ataxia, dizziness, lethargy, urticaria, pruritus.